The 3<sup>rd</sup> International Conference on Drug Discovery & Therapy: Dubai, February 7 - 11, 2011


DAY 1: Monday, February 07, 2011

3rd International Conference on

Drug Discovery & Therapy

February 7– 10, 2011, Dubai Women’s College, Dubai, UAE

www.icddt.com

 

TIME

INAUGURAL PROGRAM

09:00 -10.00 a.m.

Welcome Reception

Arrival of Participants and Guests

10.00 a.m.

Opening Ceremony

 

National Anthem

Opening Address

His Excellency Sheikh Nahayan Mabarak Al Nahayan

Minister of Higher Education and Scientific Research

Chancellor, Higher Colleges of Technology

Patron of the 3rd ICDDT

Keynote Addresses

Prof. Dr. Ferid Murad, (Nobel Laureate), Co-President, 3rd ICDDT

Prof. Dr. Atta-ur-Rahman, FRS, Co-President, 3rd ICDDT

11:00 a.m.

Coffee Break

 

COFFEE BREAK: 11:00 – 11:45 a.m.

PLENARY SESSION

Time

Chairman: F. Murad

Co-Chairman: G. Mehta

 

Speaker

Title

11:45

12:30 p.m.

Location: Auditorium

R. Huber (Nobel Laureate)
PL-1

Structure-based drug design & development with the proteasome & other intra-cellular proteases

12:30

01:15 p.m.

Location: Auditorium

E.  Neher (Nobel Laureate)

PL-2

Signals and signaling molecules in the central nervous system

01:15

02:00 p.m.

Location: Auditorium

W. Arber (Nobel Laureate)

PL-3

Molecular mechanisms of genetic variation, the driving force of biological evolution

LUNCH BREAK: 2:00 – 3:15 p.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

Hall No. 2

(First Floor)

Hall No. 3

 (First Floor)

Hall No. 4

 (First Floor)

 

Drug Delivery & Targeting/
In-Silico Drug Design & In-Silico Screening

CNS Drug Discovery & Therapy

Regenerative Medicine/Structural Biology

Hot Topics in Medicinal Chemistry

Diabetes & Obesity Drug Discovery & Therapy/Enabling Technologies

 

Chairman: J. Spencer

Co-Chairman: T. Bocan

Chairman: I. Greiner

Co-Chairman: D.P. Ramji

Chairman: H. Chao

Co-Chairman: Y.J. Woo

Chairman: I.M. Shah

Co-Chairman: V. da Silva Bolzani

Chairman: D.K. Lahiri

Co-Chairman: T.L. Peeters

03:15

03:45

p.m.

A.C. Tedesco

IL-4

Phthalocyanines derivatives loaded on liquid-crystal nanodispersions gel to skin cancer fluorescence diagnosis

03:15

03:45

p.m.

B.A. Tannous

IL-5

A novel in-vitro and in-vivo functional drug screening assay reveals lanatoside C as a potential therapeutic for glioblastoma

03:15

03:45

p.m.

M. Korbling

IL-6

Sex-mismatched stem cell transplantation: a clinical model for solid-organ tissue regeneration

03:15

03:45

p.m.

T. Yamasaki

IL-7

D-Psicose inhibits the growth of L1 stage Caenorhabditis elegans: a possible inhibition mechanism

03:15

03:45

p.m.

N.A. Khan

IL-8

A taste for fat: cell signaling mechanisms in the tongue papillae

 

03:45

04:15

p.m.

A. Coombes

IL-9

Elucidating the protein release behavior of matrix-type delivery devices using Micro-CT

03:45

04:15

p.m.

N.S. Zefirov

IL-10

Molecular design of neuroprotectors and cognition enhancers: from theory to drugs

03:45

04:15

p.m.

N. Benkirane-Jessel

IL-11

Nanostructured active biomaterials for tissue engineering applications

03:45

04:15

p.m.

P.B. Binello

IL-12

Precancerous lesions of the oral cavity: Prevention, diagnosis and cure: The state of the art

 

03:45

04:15

p.m.

T. Orban

IL-13

Autoantigen specific regulatory T cells induced in patients with type 1 Diabetes Mellitus

 

04:15

04:35

p.m.

S. Guo

SL-14

Drug-loaded multilayered films featuring uni-/dual-directional, highly adjustable, long-term sustained drug release behaviors for single-/dual-drug delivery stent application to treat malignant bodily tubular structures or cavities

 

04:15

04:45

p.m.

J. Gallinat

IL-15

In vivo cerebral glutamate monitoring in schizophrenia: Glutamate normalization in response to NMDA-receptor antagonist

04:15

04:35

p.m.

M. Bahr

SL-16

New gene therapy approaches for treatment of Parkinson’s disease

 

04:15

04:45

p.m.

T.H. Al-Tel

IL-17

Diversity oriented synthesis: synthesis, design and qualitative SAR analysis of novel anticancer motifs

 

04:15

04:35

p.m.

D.S.P. Abdalla

SL-18

Anti-inflammatory and antioxidant effects of a new arylidene-thiazolidinedione on macrophages

04:35

04:55

p.m.

A. Bouakaz

SL-19

Local drug delivery with ultrasound and microbubbles

 

04:45

05:05

p.m.

J. Feldon

SL-20

Prenatal infections and long-term mental outcome: Modeling schizophrenia-related dysfunctions using the prenatal polyl: C model in mice

 

 

04:35

04:55

p.m.

L. Calza

SL-21

Stem cells for CNS repair: alternatives to the unlikely mechanism of cell replacement

04:45

05:05

p.m.

F.B.H. Ahmad

SL-22

Enzymatic synthesis of some betulinic acid derivative: enhance their bioactivity

 

04:35

04:55

p.m.

J. Singh

SL-23

Cationic nanoparticles / nanomicelles for delivery of pDNA encoding IL-10 and pDNA encoding IL-4 and IL-10 to prevent autoimmune Diabetes

04:55

05:15

p.m.

V.B. Sulimov

SL-24

Molecular modeling in drug design: Technology and successful examples

 

05:05

05:25

p.m.

A.A. El-Rahim Abdin

SL-25

Intervention of mitochondrial dysfunction-oxidative stress-dependent apoptosis as a possible neuroprotective mechanism of alpha-lipoic acid against rotenone-induced parkinsonism and L-dopa toxicity

 

04:55

05:25

p.m.

 

IL-26

 

05:05

05:25

p.m.

H. Fallahzadeh

SL-27

HIV/AIDS Epidemic features and trends in Iran, 1986-2010

04:55

05:15

p.m.

F.Q. Parray

SL-28

Colonic J Pouch Neorectum-Is it a real gold standard?

 

 


Conference Social Mixer: 5:15 – 6:15 p.m.

The buses will leave for hotels at 6:15 p.m.


DAY 2: Tuesday, February 08, 2011

PLENARY SESSION

Time

Chairman: R. Huber

Co-Chairman: A.R. Fersht

 

Speaker

Title

09:00

09:45

a.m.

Location: Auditorium

F. Murad (Nobel Laureate)

PL-29

Application of nitric oxide research to drug development and disease therapy

09:45

10:30

a.m.

Location: Auditorium

J.-M. Lehn (Nobel Laureate)

PL-30

From supramolecular towards adaptive chemistry drug discovery aspects

 

COFFEE BREAK: 10:30 – 11:15 a.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

 

Hall No. 3

 (First Floor)

 

Hall No. 4

 (First Floor)

 

 

Drug Delivery & Targeting/
Anti-Cancer Drug Discovery & Therapy

CNS Drug Discovery & Therapy

Cardiovascular Drug Discovery & Therapy

Enabling Technologies/Hot Topics in HIV Research

 

Recent Advances in Patient Treatment & Care

 

Chairman: N.A. Darmani

Co-Chairman: P. Srinivas

 

Chairman: B.A. Tannous

Co-Chairman: N. Zefirov

Chairman: M.F.A. Adamo

Co-Chairman: N. Benkirane-Jessel

Chairman: T. Yamasaki

Co-Chairman: P. Nemani

Chairman: J.G. Zayas

Co-Chairman: E. Terpos

11:15

11:45

 a.m.

Y. Tamaki

IL-31

Novel nanotechnology-based drug delivery in photodynamic therapy for age-related macular degeneration

11:15

11:45

 a.m.

I. Greiner

IL-32

Cariprazine, an antipsychotic PIII compound

 

11:15

11:45

 a.m.

D.P. Ramji

IL-33

The macrophage foam cell as a promising therapeutic target for atherosclerosis

11:15

11:45

 a.m.

P. Stadler

IL-34

Robot-assisted Vascular Surgery

11:15

11:45

 a.m.

R.-P. Mueller

IL-35

The successful coordination of chemo- and radiotherapy to optimize outcome and toxicity in early stages Hodgkin’s Lymphoma.  The final results of the HD-10 trial of the German Hodgkin study group with 1370 patients

 

11:45

12:15

p.m.

 

IL-36

 

11:45

12:15

p.m.

W. Jia

IL-37

Innovative approaches for a novel antidepressant from traditional Chinese medicine

 

11:45

12:15

p.m.

Y.J. Woo

IL-38

Mathematically designed synthetic polypeptide analog of stromal cell-derived factor 1 alpha functions as a superpotent neovasculogenic agent for treating myocardial ischemia

 

 

 

 

11:45

12:15

p.m.

S. Stahl

IL-39

Affibody technology targeting cancer and Alzheimer’s disease

 

11:45

12:15

p.m.

R.L. Jones

IL-40

Advances in the systemic management of sarcomas

 

12:15

12:45

p.m.

B. Fang

IL-41

Developing novel multipathway modulating anticancer agents

12:15

12:45

p.m.

S. Bellino

IL-42

Recent advances in treatment of borderline personality disorder (BPD)

 

12:15

12:45

p.m.

H. Tomoda

IL-43

In-vivo efficacy of pyripyropene derivatives in atherogenic mouse models

 

12:15

12:45

p.m.

M. Koffas

IL-44

Engineering plant secondary metabolite biosynthesis in microorganisms

 

12:15

12:45

p.m.

T.L. Peeters

IL-45

How to let patients benefit of motilides: A new approach

 

12:45

01:15

 p.m.

S.A. Grando

IL-46

Anti-Tumorigenic effects of small cholinergic peptides of the LY6 protein family

 

12:45

01:15

 p.m.

Y. Tanaka

IL-47

Aphasia, anxiety, and beta-adrenergic antagonists

 

12:45

01:15

 p.m.

F.A. Villamena

IL-48

Development of new spin traps for therapeutics

 

12:45

01:15

p.m.

R. Di Santo

IL-49

Diketo acids derivatives as dual inhibitors of human immunodeficiency virus type 1 integrase and the reverse transcriptase RNase H Domain

12:45

01:15

 p.m.

A. Di Pietro

IL-50

Targeting the multidrug resistance-conferring ABC transporters overexpressed in cancer cells: in-vitro optimization and in-vivo validation

 

01:15

01:45

p.m.

 

IL-51

 

01:15

01:45

p.m.

Y. Iwasaki

IL-52

Trophic effect of olmesartan on spinal motor neurons in vitro and in vivo

 

01:15

01:45

p.m.

A.J. Merched

IL-53

Vascular inflammation: Light at the end of the tunnel

 

01:15

01:45

p.m.

M. Peterlin

IL-54

HIV latency and HDAC inhibitors

01:15

01:35

p.m.

C.S. Ulrik

SL-55

Management of Asthma in pregnancy

 

LUNCH BREAK: 01:45 – 02:45 p.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

 

Hall No. 3

 (First Floor)

 

Hall No. 4

 (First Floor)

 

 

Anti-Cancer Drug Discovery & Therapy/Stereoselective Synthesis of Bioactive Compounds

Medical Imaging

Inflammation & Immunology

Hot Topics in Natural Products

Diabetes & Obesity Drug Discovery & Therapy/
High-Throughput Screening & Laboratory Automation

 

 

Chairman: B. Fang

Co-Chairman: A. Albini

Chairman: S. Bellino

Co-Chairman: Y. Tanaka

Chairman: P.C. Heinrich

Co-Chairman: F.A. Villamena

Chairman: P.B. Binello

Co-Chairman: O. Hammarsten

Chairman: N.A. Khan

Co-Chairman: D.S.P. Abdalla

 

02:45

03:15

p.m.

U. Manne

IL-56

Effect of pre-clinical research on cancer disparities to evidence-based care

 

02:45

03:05

p.m.

A. Benabarre

SL-57

The correlation of cerebral blood flow and neuropsychology in bipolar patients

 

02:45

03:05

p.m.

S.Y. Seong

SL-58

Agonist for G-protein coupled receptor 131 attenuate systemic inflammatory syndrome

 

02:45

03:05

p.m.

R.D. Lele

SL-59

Chemoprevention of cancer

 

02:45

03:05

p.m.

M.A. Leissring

SL-60

Designed inhibitors of insulin-degrading enzyme as promising pharmacophores for the treatment of diabetes

 

03:15

03:35

p.m.

P. Srinivas

SL-61

Multifaceted approach with a single drug for BRCA1 defective cancers

 

03:05

03:25

p.m.

F. Pilleul

SL-62

CT scan in colonic cancer as a screening test

 

03:05

03:25

p.m.

A.I. Tchorbanov

SL-63

Experimental therapy in humanized SCID mice models of SLE

 

 

03:05

03:25

p.m.

D. de F. Buchi

SL-64

M1 as a promising product that modulates NF-kB activation

03:05

03:25

p.m.

D. Li

SL-65

Fibroblast growth factor-21 ameliorates both diabetes and obesity

03:35

03:55

p.m.

S. Gou

SL-66

Biological evaluation of novel structure-activity platinum complexes

 

03:25

03:45

p.m.

Y. Ni

SL-67

Medical imaging research leads to discovery of a new anticancer strategy

03:25

03:45

p.m.

J. Vojinovic

SL-68

First use of oral histone deacetylase inhibitor (Givinostat) in systemic Onset Juvenile Idiopathic Arthristic (Sojia)

03:25

03:45

p.m.

E.V. Soniya

SL-69

A novel polyketide synthase from ginger – a prime candidate for natural medicinal compound biosynthesis

 

03:25

03:45

p.m.

F. Samad

SL-70

Targeting de novo ceramide biosynthesis ameliorates multiple features of the metabolic syndrome in diet induced obesity

03:55

04:15

p.m.

N.A. Darmani

SL-71

A re-evaluation of the neurochemical and anatomical bases of chemotherapy-induced vomiting

03:45

04:05

p.m.

M. Chorazy

SL-72

Histopathological diagnosis of small cell lung cancer through the biopsy of spleen metastases under ultrasound examination

 

03:45

04:05

p.m.

J.N. Agrewala

SL-73

Caerulomycin A: A novel immunosuppressive agent that modulates the activity of both T cells and B cells

03:45

04:05

p.m.

M.A. O’Neil-Johnson

SL-74

High-throughput natural products chemistry for drug discovery: Is it possible?

03:45

04:15

p.m.

J.G. Bueno

IL-75

Antimicrobial drug discovery, screening predicts the clinical outcome?

04:15

04:35

p.m.

J.K. Ray

SL-76

Use of “halo vinyl aldehydes” in organic synthesis and chemo selective functional group transformations in gamma lactam derivatives

 

04:05

04:25

p.m.

W.A. Zaghary

SL-77

Labeling and biodistribution of 99mTc-7-Bromo-1, 4-dihydro-4-oxo-quinolin-3-carboxylic acid complex

04:05

04:25

p.m.

L.Y. Al-Ayadhi

SL-78

Serum levels of brain-derived neurotrophic factor (BDNF) in autistic children

04:05

04:25

p.m.

P.M. Sherief

SL-79

Extraction, characterization, antioxidant property and anti-inflammatory activity of carotenoids from the shell waste of Arabian red shrimp Aristeus alcocki (Ramadan, 1938)

 

04:15

04:35

p.m.

Y.-T. Chang

SL-80

Development of bioimaging probes for in-vitro, in-vivo and clinical applications by diversity oriented fluorescence library approach (DOFLA)

 

POSTER PRESENTATION: 04:25 – 6:00 p.m.


Posters Session: 4:25 – 6:00 p.m. at corridor

Gala Dinner at Dhow Cruise: Departure at 6:00 p.m.

The buses will leave for hotels at 8:30 p.m.


DAY 3: Wednesday, February 09, 2011

PLENARY SESSION

Time

Chairman: E. Neher

Co-Chairman: T. Bocan

 

Speaker

Title

09:00

09:45

a.m.

Location: Auditorium

G. Mehta

PL-81

Probing synergy between natural products and total synthesis for human wellbeing

 

09:45

10:30

a.m.

Location: Auditorium

Sir A.R. Fersht

PL-82

The tumour suppressor p53: From structure to drug discovery

 

COFFEE BREAK: 10:30 – 11:15 a.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

 

Hall No. 3

 (First Floor)

 

Hall No. 4

 (First Floor)

 

Hall No. HS-1008

(Ground Floor)

 

 

Hot Topics in Drug Targets

Drug Discovery in Preclinical Research

Proteomics & Bioinformatics/
Pharmaceutical Research & Development

Pharmacogenomics/
Translational Medicine

 

Hot Topics in Natural Products/Recent Advances in Patient Treatment & Care

 

Academic CRO/Industrial Collaborations in Drug Discovery

 

Chairman: B. Stefanovic   Co-Chairman: J. Vojinovic

 

Chairman: Taleb Al-Tel

Co-Chairman: M.A. Leissring

Chairman: G.H. Scherr

Co-Chairman: Prathima Srinivas

 

Chairman: S.Y. Seong

Co-Chairman: N. Benkirane-Jessel

Chairman: I. Toth

Co-Chairman: A. Kocak

Chairman: A. Al Amiri

Co-Chairmen: M. Al-Farhan /K. Kodukula

11:15

11:45

a.m.

P. Nemani

IL-83

Targeting gp96 to prevent neonatal meningitis

11:15

11:45

a.m.

M.I. Choudhary

IL-84

Productivity crises in pharmaceutical sector – Nature’s Answer

 

11:15

11:45

a.m.

I.H. Khan

IL-85

Phosphoproteomic profiling of signaling pathways in cancer cells by microparticle suspension arrays

 

 

11:15

11:45

a.m.

I.M. Shah

IL-86

Antithrombotic therapy and cytochrome P450 pharmacogenomics

 

 

 

11:15

11:45

a.m.

O. Hammarsten

IL-87

Repeated transient sulforaphane stimulation in astrocytes leads to prolonged Nrf2-mediated gene expression and protection from superoxide-induced damage

 

11:15

12:15

p.m.

R. Chaguturu

SIL-88

Current trends in collaborative drug discovery and strategies to De-risk open innovation-based precompetitive initiatives

 

11:45

12:15

 p.m.

G. Sansoe

IL-89

Portal hypotensive action of calcimimetic agents in rats with Ccl4-induced ascitic liver cirrhosis

11:45

12:15

 p.m.

D.K. Lahiri

IL-90

Discovery of a novel drug target for Alzheimer’s disease: miR-101 regulates levels of the amyloid precursor protein

 

11:45

12:05

 p.m.

R. Issa

SL-91

Identification of glucosinolate QTLs in Brassica oleracca C genome revealed interesting genome regions for biological applications

 

11:45

12:05

 p.m.

A. Lezhava

SL-92

Rapid detection of clinically important SNPs and mutations by two-color SmartAmp method

 

 

 

 

11:45

12:15

 p.m.

V. da Silva Bolzani

IL-93

Will natural chemistry diversity from tropical biodiversity continue to inspire medicinal chemistry?

12:15

12:45

p.m.

L. Lafanechere

IL-94

A new pharmacological inhibitor of LIM Kinase that blocks cell motility and stabilizes microtubules

12:15

12:45

p.m.

M.D. Hamalainen

IL-95

The importance of drug-target binding kinetics for drug efficacy – Without on you are off!

12:05

12:25

p.m.

T. Shah

SL-96

The use of proteomics and bioinformatics to develop a serum based diagnostic test for feline lymphoma

 

12:05

12:35

p.m.

C.J. Henry

IL-97

Use of spontaneously arising canine TCC as a relevant model of late-stage human bladder cancer in which to assess the novel drug, Tavocept TM, for its ability to mitigate toxicity and improve efficacy of a cisplatin and piroxicam combination therapy protocol

 

12:15

12:45

p.m.

M.-T. Liong

IL-98

Cholesterol-reducing effects of a symbiotic containing Lactobacillus acidophilus and inulin in hypercolesterolemic subjects

 

12:15

12:45

p.m.

W.R. Hume

IL-99

Productive government, university and industry relationships in research

 

12:45

01:05

p.m.

N.V. Koshkina

SL-100

The Fas mechanism as a novel target to treat lung metastases using metastatic osteosarcoma model

12:45

01:05

p.m.

F. Vyskocil

SL-101

Alkylammonium derivatives of 6-methyluracil act as tissue-specific inhibitors of acetylcholine esterases in muscle and brain

 

12:25

12:45

p.m.

T. Comoglu

SL-102

Formulation technologies & future research trends of orally fast disintegrating Tablets

12:35

01:05

p.m.

P. Bernardi

IL-103

Toward a mitochondrial therapy of muscular dystrophies: From mouse model to clinical trial

 

12:45

01:15

p.m.

J. Schripsema

IL-104

Metabolomics in the discovery of novel drugs

 

12:45

01:05

p.m.

N. Sulaiman

SL-105

Academia-industry collaboration in training and research – the Sharjah model

 

 

01:05

01:25

p.m.

P. Trapencieris

SL-106

New selective CA-I inhibitors

 

01:05

01:25

p.m.

R.J. Anto

SL-107

Chemosensitizing efficacy of curcumin in paclitaxel chemotherapy as evidenced by chemical-induced and xenograft models of cervical cancer

 

12:45

01:05

p.m.

G. Shahnaz

SL-108

Intestinal lymphatic drug delivery of phenothiazines by ex-vivo model: Influence of self-nanoemulsifying formulation design 

 

01:05

01:25

p.m.

V.N. Smirnov

SL-109

Cord blood cells (CBC) in the treatment of brain trauma and cerebral palsy

 

01:15

01:35

p.m.

E. Terpos

SL-110

The role of antiresorptive agents in the management of multiple myeloma-related bone disease

01:05

01:25

p.m.

O. Shafey

SL-111

Regulation and promotion of health research in Abu Dhabi

 

01:05

01:25

p.m.

S. Danti

SL-112

Middle Ear Tissue Engineering: new challenges and opportunities for otologic surgery

 

 

 

LUNCH BREAK: 01:25 – 2:30 p.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

 

Hall No. 3

 (First Floor)

 

Hall No. 4

 (First Floor)

 

Hall No. HS-1008

(Ground Floor)

 

 

Inflammation & Immunology/Hot Topics in Drug Targets/Innovative Drug Discovery & Nanotechnology

Recent Advances in Spectroscopy/ Proteomics & Bioinformatics

 

Anti-Infectives/Hot Topics in Medicinal Chemistry

 

Hot Topics in Natural Products

Recent Advances in Patient Treatment & Care

Academic CRO/Industrial Collaborations in Drug Discovery

 

Chairman: L. Lafanechere

Co-Chairman: G. Sansoe 

Chairman: I.H. Khan

Co-Chairman: D.K. Lahiri

Chairman: F. Pilleul

Co-Chairman: Y. Ni

 

Chairman: M.T. Liong

Co-Chairman: R.D. Lele

Chairman: R.L. Jones

Co-Chairman: H. Chao

Chairman: R. Chaguturu

Co-Chairman: K. Kodukula

 

02:30

03:00

p.m.

 P.C. Heinrich

IL-113

Pro-inflammatory cytokines impair IL-6 mediated STAT3 activation by serine phosphorylation and subsequent internalization of the signal transducer gp130

02:30

03:00

p.m.

A. Kocak

IL-114

The role of vibrational spectroscopy in modern forensic science research

 

02:30

03:00

p.m.

G.H. Scherr

IL-115

Instant hand sanitizers

 

02:30

03:00

p.m.

M.A. O’Neil-Johnson

IL-116

New chemical scaffold starting points for targeting inflammation preferred, novel and neglected scaffolds in a drug discovery program

 

02:30

03:00

p.m.

D. Martin

IL-117

Intraoperative radiation therapy: Past, present & future

 

 

 

02:30

03:00

p.m.

S. Herzig

IL-118

Graduate program in pharmacology and experimental therapeutics – a joint endeavor of the University of Cologne and Bayer Schering

 

03:00

03:30

 p.m.

A.M. Artoli

IL-119

Mechanism of inflammation: A simulation approach

 

03:00

03:20

p.m.

A. Freiberg

SL-120

Membrane proteins under high hydrostatic pressure reveal cooperative and reversible rupture of hydrogen bonds

 

03:00

03:20

 p.m.

M. Mares

SL-121

In vitro activity of a novel propiconazole derivative (MXP-4509) nanoparticle-formulated

03:00

03:20

 p.m.

K.W. Wellington

SL-122

A Laccase-catalysed synthesis of naphthoquinone Bis-Sulfides

03:00

03:20

 p.m.

L. Moezi

SL-123

The effect of pioglitazone, a specific ligand of the proxisome prolifrator-activated receptor gamma, on ethanol - induced gastric ulcers in cirrhotic rats: The role of nitric oxide and IL1-β

 

 

 

 

 

 

 

 

 

 

 

03:00

03:30

 p.m.

W. Moos

IL-124

Nonprofit pharma

 

03:30

03:50

p.m.

A.Y. Ozer

SL-125

Investigating cold chain system and efficacy of vaccines that have reached to the market in Turkey and related legal provisions

 

03:20

03:40

p.m.

A.K. Gajjar

SL-126

Impurity profiling: A case study of ezetimibe

03:20

03:40

p.m.

J. Tazi

SL-127

Therapeutic modulation of HIV-1 alternative splicing by small molecules: A novel strategy for AIDS treatment

03:20

03:40

p.m.

B.H. Jacobson

SL-128

Efficacy of two concentrations of comfrey root (symphytum officinale L.) extract ointments combined with tannic acid in the treatment of patients with primary osteoarthritis of the knee: A double-blind, randomized, multicenter, placebo-controlled trial

 

03:20

03:40

p.m.

J. Lipozencic

SL-129

Toxic epidermal necrolysis with fatal outcome by lansoprasole

03:30

03:50

p.m.

Assem S. el Baghdady

SL-130

Unlocking the market potential of academic research

 

03:50

04:10

p.m.

B. Stefanovic

SL-131

A novel target for antifibrotic drugs and a high throughput assay to screen for such drugs

03:40

04:00

p.m.

M. Claybourn

SL-132

Technology and scientific advancements that will lead to further improvements in understanding drug behavior

 

03:40

04:00

p.m.

C.O.Rangel-Yagui

SL-133

Micellar partition coefficient of drugs as a parameter to estimate blood-brain barrier penetration

 

03:40

04:00

p.m.

K. Awang

SL-134

The Malaysian flora, a rich source of lead compounds

 

03:40

04:00

p.m.

J.G. Zayas

SL-135

Developing a new paradigm in respiratory hygiene to control transmission of infectious respiratory diseases and to optimize respiratory secretions management

 

03:50

04:10

p.m.

G. AlTajir

SL-136

Regulatory requirements in collaborative research

 

04:10

04:30

p.m.

B. Chen

SL-137

Ginkgolide B inhibition of the inflammatory protein expression associated with reduce NOX4 expression and NF-κB activation in ox-LDL-stimulated HUVECs

04:00

04:20

p.m.

H. Lamela

SL-138

New laser optoacoustic spectroscopy (LOS) system to quantify gold nanoparticles in a liquid tissue phantom for biomedical applications

04:00

04:20

p.m.

Zia-ur-Rehman

SL-139

Structural properties, antimicrobial and anticancer potency of new organotin(IV) dithiocarboxylates

04:00

04:20

p.m.

F. Maiza-Benabdesselam

SL-140

Antibacterial activity of essential oils of two Algerian medicinal plants orignum glandulosum Desf.  And Artemisia herba alba Asso

04:00

04:20

p.m.

M.B. Jakovljevic

SL-141

Anticonvulsant plasma concentration impact on seizure control, life quality and drug adverse events in teenagers and adult youths with epilepsy

 

 

 

04:10

04:30

p.m

A.M. Al-Ghananeem

SL-142

Challenges in parenteral dosage from preparations of slightly water-soluble drugs: dantrolene sodium’s successful example of academic-industrial collaboration

04:30

04:50

p.m.

B. Azizi

SL-143

GFP chromophores as potential ligands for the estrogen receptor and the pregnane X Receptor

04:20

04:50

p.m.

H. Durchschlag

IL-144

Prediction of discrete water molecules preferentially bound to proteins and of water channels in protein interiors

 

04:20

04:40

p.m.

A. Badshah

SL-145

DNA binding potency of new ferrocenyl amides

 

04:20

04:40

p.m.

S.M. Adekenov

SL-146

Prospects of development of new preparations on the basis of natural sesquiterpene lactones

04:20

04:50

p.m.

C.D. Ribas

IL-147

Long-Term effects of long-acting beta 2-agonists: What the literature tells and doesn’t tell us

 

04:30

04:50

p.m

Yazeed A Al-Sheikh

SL-148

Assessing inborn errors of metabolism in Saudi Arabia and improved methods of screening and diagnosis

POSTER PRESENTATION: 04:40 – 6:00 p.m.


Posters Session: 4:40 – 6:00 p.m. at corridor

Shopping Tour: Departure at 6:00 p.m.



DAY 4: Thursday, February 10, 2011

PLENARY SESSION

Time

Chairman: W. Arber

Co-Chairman: D.K. Lahiri

 

Speaker

Title

09:00  09:45

a.m.

Location: Auditorium

T. Bocan

PL-149

 

Application of platform imaging biomarkers in drug discovery - focus on neuroscience, oncology and cardiovascular

 

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

Hall No. 3

 (First Floor)

Hall No. 4

 (First Floor)

Hall No. HS-1008

(Ground Floor)

 

 

Diabetes & Obesity Drug Discovery & Therapy

 

Stereoselective Synthesis of Bioactive Compounds/ Enabling Technologies

Pharmaceutical Research & Development

Cardiovascular Drug Discovery & Therapy

Innovative Drug Discovery & Nanotechnology

Protein & Peptide Sciences

 

Chairman: R.J. Anto

Co-Chairman:

F. Vyskocil

Chairman: B.H. Jacobson

Co-Chairman: J.K. Ray 

Chairman: M.A. O’Neil-Johnson

Co-Chairman: J. Tazi

Chairman: F. Huq

Co-Chairman: M.D. Hamalainen

Chairman: J.G. Zayas

Co-Chairman: R.L. Jones

Chairman: M.I. Choudhary

Co-Chairman: D.K. Lahiri

 

09:50

10:20

a.m.

S. V. Karnataki

IL-150

Diabetes and obesity drug discovery and therapy

09:50

10:20

a.m.

M.F.A. Adamo

IL-151

Novel synthetic methodologies to prepare unnatural acids, aminoacids and peptidomimetics

 

09:50

10:20

a.m.

V.I. Perez-Nueno

IL-152

Predicting drug polypharmacology by correlating ligand and target shape similarities

 

09:50

10:20

a.m.

S.D. Bergese

IL-153

Perioperative blood pressure control, is clevidipine the answer?

09:50

10:20

a.m.

T. Moos

IL-154

Gene delivery by pullulan derivatives in brain capillary endothelial cells for protein secretion

09:50

10:10

a.m.

T. Santos-Silva

SL-155

CORM-3 Reactivity towards proteins: The crystal structure of a Ru(II) Dicarbonyl-Lysozyme complex

 

10:20

10:40

a.m.

C.-H. Chou

SL-156

Hypoglycemic natural products of cucurbitaceae-type triterpenoids from plants of the cucurbitaceae family

 

10:20

10:40

a.m.

H.A. Al Attar

SL-157

Monitoring the emergence of drug resistance in patients treated with imatinib (GlivecR) by identifying SNP in ABL portion of the BCR-ABL oncogene using fluorescence method

 

10:20

10:40

a.m.

A. Alfaki

SL-158

Cardiac neurons firing precedes cortical neurons firing by variable time equivalent to RP or Lipet’s latency period in goal directed behavior or action in conscious state

10:20

10:40

a.m.

K. Smiljanic

SL-159

Involvement of MMP-2 and ADAM-12 in thrombin-induced rat’ VSMCs proliferation

 

10:20

10:40

a.m.

M.V. Khvostov

SL-160

The improvement of toxico-pharmacological properties of drugs by clathration with plant metabolities

10:10

10:30

a.m.

B. Kundu

SL-161

A novel thermostable L-asparaginase with a promising anti-cancer activity

 

OFFEE BREAK: 10:40 – 11:10 a.m.

 

Lecture Hall

(Ground Floor)

Multipurpose Hall

 (Hall 1 - First Floor)

 

Hall No. 2

(First Floor)

 

Hall No. 3

 (First Floor)

 

Hall No. 4

 (First Floor)

 

Hall No. HS-1008

(Ground Floor)

 

 

Anti-Cancer Drug Discovery & Therapy/ Drug Delivery & Targeting

Regenerative Medicine/ Pulmonary Drug Discovery & Therapy

 

Diabetes and Obesity Drug Discovery & Therapy/

Cardiovascular Drug Discovery & Therapy/ Oncology

Recent Advances in Patient Treatment & Care

Biologics/In-Silico Drug Design & In-Silico Screening

Drug Discovery in Preclinical Research/Combinatorial Chemistry/ Innovative Drug Discovery & Nanotechnology/ Pharmaceutical Biotechnology

 

Chairman: V.I. Perez-Nueno

Co-Chairman: G. Shahnaz

 

Chairman: M.I. Choudhary

Co-Chairman: A. Kocak

Chairman: T. Moos

Co-Chairman: M.V. Khvostov

Chairman: R.H. Davies

Co-Chairman: A. Di Pietro

Chairman: M.F.A. Adamo

Co-Chairman: R. Pasqualini

 

Chairman: D. Li

Co-Chairman: M.-T. Liong

11:10

11:40

a.m.

F. Huq

IL-162

Synergism from combinations of platinums with phytochemicals as applied to ovarian cancer

 

11:10

11:40

a.m.

A. Al-Hendy

IL-163

Adenovirus-mediated overexpression of human tissue plasminogen activator prevents peritoneal adhesion formation/reformation

 

11:10

11:40

a.m.

K. Miyashita

IL-164

cGMP-dependent protein kinase cascades increase muscle mitochondrial content and prevent obesity and diabetes

11:10

11:40

a.m.

M.R. El-Gewely

IL-165

CCMP, a new road for the treatment of monogenic diseases due to mutations; its use on chemo-resistant cancers

11:10

11:40

a.m.

S. Dubel

IL-166

Human antibody – Human RNase fusion proteins for tumor therapy

 

11:10

11:40

a.m.

J.N. Bryan

IL-167

Use of spontaneously arising canine lymphoma as a preclinical model of DNA methylation derangements for drug target identification

 

11:40

12:10

p.m.

G. Birkenmeier

IL-168

How to command the wnt/B-cantenin pathway from outside of the tumor cell: the A2M-LRP1 axis

 

11:40

12:00

noon

J.A. Andrades

SL-169

Articular cartilage regeneration by autologous mesenchymal stem cells using a novel nano-composite collagenous scaffold

 

11:40

12:10

p.m.

K.C. Norris

IL-170

A novel cystine based antioxidant attenuates high fat diet-induced oxidative stress and hepatic steatosis in apoliporotein E knockout mice

 

11:40

12:10

p.m.

H. Chao

IL-171

L-DOS47 – A phase I/II lung cancer candidate that uses tumor alkalization as a therapeutic approach

 

11:40

12:10

p.m.

M.F. Bachmann

IL-172

Targeting plasmocytoid dendritic cells with protein-based nanoparticles for the treatment of asthma

11:40

12:10

p.m.

J. Spencer

IL-173

Parallel synthesis of libraries of medicinal interest

12:10

12:30

p.m.

J.M. Moshi

SL-174

The effects of UV solar light radiation on live cells using yeast (Saccharomyces cerevisiae) as a model of eukaryotes

 

12:00

12:20

p.m.

L.M. Popescu

SL-175

Telocytes and stem cells: a tandem in cardiac regenerative medicine

 

12:10

12:30

p.m.

M. Sharma

SL-176

Evaluation of antidiabetic and antioxidant effects of Seabuckthorn (Hippophae rhamnoides L.) in streptozotocin-nicotinamide induced type-2 diabetic rats

 

 

 

 

 

12:10

12:40

p.m.

V.D. Garovic

IL-177

Podocyturia in patients treated with VEGF blocking therapy for cancer

 

 

12:10

12:30

p.m.

M.R. El-Gewely

SL-178

Early-stage hurdles in recombinant therapeutics development and the impact of our novel Conformases/Foldases

12:10

12:30

p.m.

L. Saleh

SL-179

Selenopeptide phage display: Chemical modification and applications

 

12:30

01:00

p.m.

I. Toth

IL-180

Multi-epitopic vaccine delivery system: Synthesis and investigation

 

12:20

12:40

p.m.

 

SL-181

 

12:30

12:50

p.m.

P. Cervinka

SL-182

Optical coherence tomography guided primary PCI in STEMI patients.  A pilot study 

 

12:40

01:00

p.m.

R. Turner

SL-183

Plasma coating – Meeting the Hfa challenge, the latest in can Technology is here

 

12:30

01:00

p.m.

 

IL-184

 

12:30

01:00

p.m.

S.S. Farber

IL-185

A new approach to the design and synthesis of drugs based on self-organizing quasi-life systems

 

01:00

01:20

 p.m.

N.E. Polyakov

SL-186

Water soluble drugs conjugates with oligo- and polysaccharides.  New approach for drug design and delivery

12:40

01:00

 p.m.

M.S. Kannan

SL-187

Role of CD38 in Asthma

 

12:50

01:10

p.m.

A. Kopylov

SL-188

Novel modular DNA aptamer for human thrombin with high anticoagulant activity

 

01:00

01:20

p.m.

N. Arslani

SL-189

Advantages of new materials in fascia transversalis reinforcement for inguinal hernia repair

 

01:00

01:20

p.m.

V. Ramakrishnan

SL-190

A ‘reductionist’ approach in virtual activity profiling of drug molecules

 

01:00

01:20

p.m.

P. Srinivas

SL-191

Acyclovir loaded solid lipid nanoparticulate systems – Formulation, characterization and pharmacokinetic evaluation for oral and parenteral routes

 

01:20

01:40

p.m.

Anmin Li

SL-192

Magnetic paclitaxel nanoparticles inhibit glioma growth and improve the survival of rats bearing glioma xenografts

 

 

01:00

01:20

p.m.

P.A. Singleton

SL-193

High molecular weight hyaluronan is a novel inhibitor of acute lung injury

 

01:10

01:30

p.m.

S. Sirpal

SL-194

Injury, infection, and inflammation – The trilogy of vascular disease

01:20

01:40

p.m.

M. Kabir-Salmani

SL-195

Properties of L-type amino acid transporter 1 (LAT1) in epidermal ovarian cancer

01:20

01:40

p.m.

M. El-Hefnawi

SL-196

Computer-Aided drug design and drug discovery efforts for hepatitis C virus: Novel polymerase inhibitors and optimal small interfering RNAs targeting the HCV genome

 

01:20

01:40

p.m.

Z. Zakaria

SL-197

In-vitro production of antioxidants of naringin and hesperidin and their activity in unsaturated fatty acid for oil preparation pharmaceuticals

 

 

01:40

02:00

p.m.

B. El-Gamal

SL-198

New trends in drug delivery and targeting: Potential clinical applications

 

01:20

01:40

p.m.

S. Rao

SL-199

Levofloxacin in retreatment of Pulmonary Tuberculosis – An experience with twenty patients

 

01:30

01:50

p.m.

A.B.M.F. Karim

SL-120

Chemotherapy induced thrombocytopenia for solid cancer and lymphoma: A novel herbal solution

 

01:40

02:00

p.m.

C.D. Ribas

SL-201

Omalizumab effect in non-allergic asthma patients

01:40

02:00

p.m.

A. Nandy

SL-202

Multational patters in avian and swine flue viruses and identification of surface exposed conserved region in neuraminidase and VP7 proteins by graphical representation and numerical characterization (granch) studies

 

01:40

02:00

p.m.

A. Grammenos

SL-203

A combination of ESR and SANS techniques to explore the Cyclodextrin action on membranes

 

01:40

02:00

p.m.

S.O. Arslan

SL-204

Evaluation by in vivo respiration enrolled of lung toxicity in rats kept in coal mine ambience: effect of antioxidant therapy

 

02:00

02:20

p.m.

H.G. Abdelhady

SL-205

4Dimensions atomic force microscopy investigation of the packing and un-packing of dendritic-DNA nanoplexes

LUNCH BREAK: 02:00 – 03:15 p.m.

POSTER PRESENTATIONS: 03:15 – 4:15 p.m.

CASH PRIZE ANNOUNCEMENT FOR THREE BEST POSTERS: 4:15 p.m.

POSTER PRESENTER’S PRESENCE IS ESSENTIAL TO RECEIVE THE CASH AWARD AND CERTIFICATE OF MERIT

Posters Session: 03:15 – 4:15 p.m.

City Tour: Departure at 4:20 p.m.

 

IMPORTANTThe buses will leave daily from all Hotels at 8:15 a.m. for the conference venue. 

 

PL: Plenary Lecture

SIL: Special Invited Lecture

IL: Invited Lecture

SL: Session Lecture

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