Name of Speaker |
Title |
P. Boulikas |
Tumor-Targeted
Liposomal Cisplatin (Lipoplatin™) and Oxaliplatin
(Lipoxal™) show Superiority to Free Drugs: from
Inception to Phase III |
G. Campiani |
Development
of Potent Atypical Antipsychotics based on A Novel Neurochemical
Approach |
P. Talaga |
Frontiers
in Medicinal Chemistry. Time for another Big Bang? |
N. Pugno |
Smart
Flexible Nanovectors |
G. Osuji |
Discovery
of the RNA Synthetic Activity of Glutamate Dehydrogenase
and Application in Drug Metabolism |
A.D.N. Vaz |
Aldehyde
Oxidase in Drug Metabolism: Simple Preclinical Tests to
Avoid Potential for Clinical Pharmacokinetic Failure |
A. Milosavljevic |
A
Comprehensive Map of Chromosomal Aberrations in the MCF-7
Breast Cancer Cell Line Genome: Technology, Informatics,
and Significance |
F.M. Veronese |
Therapeutic
Proteins: New Achievements for Stabilization and Delivery |
B. Roca (Villanueva) |
Pharmacogenomics
of Antiretrovirals |
D. Grainger |
Title Awaited
|
P.G.M. Rao |
Adverse
Drug Reactions among Hospitalized Patients in Nephrology
Wards-An Intensive Monitoring Study |
K. Yasuda |
Title Awaited
|
K.K.W. Wang |
New
Theranostic Approach to Diagnose and Treat Traumatic Brain
Injury |
R. Minchin |
Multi-Component
Peptide-Based Carriers for Non-Viral DNA Delivery |
F. Darvas |
Enabling
Novel Technologies to Expedite Medicinal Chemistry: Combination
of Flow Synthesis and Serendipity-Enhancing Technics for
Lead D iscovery |
Y. Perrie |
Delivering
DNA and Protein Antigens – A Role For Cationic Liposomes |
P. Simerska |
Vaccines
against group A Streptococcal Infection and Human Papillomavirus
Type-16 associated Cervical Cancer |
M. Stenzel |
Crosslinked
Micelles via the Raft Process: Towards a more Biocompatible
Gene Delivery System |
E. Gordon |
Integrating
Gene-Brain-Behaviour Markers for the era of ‘Personalized
Medicine’ |
E. Kmonickova |
Nitric
Oxide as a Biomarker of Immunostimulatory Activity of
Drugs |
Y. Korpan |
Cancer
Diagnostic and Prognostic: European Research Strategies,
Recent Sensor Achievements and New Targets |
R. McDade |
Following
the Critical Path: Development of Multi-Analyte Profiles
for Sensitive, Early Detection of Toxicity |
S. Mukaddam-Daher |
Cardiac
Imidazoline Receptors, a New Therapeutic Target |
K.S.A. Khabar |
Molecular
Response to Therapeutic Interferons: Sensitivity and Resistance
Mechanisms |
M. Yoshioka |
Identification
and Characterization of Therapeutic Targets for Prostate
Cancer |
B. Rochat |
Role
and Importance of Hepatic and Extrahepatic Drug Metabolizing
Enzymes in the Bioavailability of Anti-Cancer Agents in
Cancer Cells |
V. Apostolopoulos |
Peptide
based Vaccines: A Structural and Immunological Perspective |
U. Bachrach |
Imino-aldehydes-
a new tool to Combat Cancer and Viral Diseases |
U. Baltayev |
Antiulcer
and Cardiovascular Compounds(steroids): Structure Activity |
A.J. Mendonca |
Novel
Building Blocks and Templates for GPCR and Kinase Research |
C. Maercker |
Inducible
Nidogen Expression in Epidermal HACAT Cells |
J. Nielsen |
Synthesis
of Bioactive Natural Products |
V. Sakanyan |
Development
of Small Molecule and Antibody Microarrays Designed for
Drug Discovery |
In-C. Kang |
High-Performance
Screening of Active Peptide Inhibitor of Integrin Receptor
by Protein Microarray Chip |
J. Tavernier |
The
MAPPIT Toolbox: Strategies to Analyze Molecular Interactions
in Intact Cells |
A. Yuryev |
In
Silico Pathway Analysis: The Final Frontier Towards Completely
Rational Drug Design |
S. Hannongbva |
Title Awaited |
J. Turnbull |
“Engineered
Heparins”: Novel Beta-Secretase Inhibitors as Potential
Therapeutics for Alzheimer's Disease |
B. Potter |
Steroid
Sulfatase Inhibitors: From Concept to Clinic |
A. Tsarbopoulos |
Title Awaited |
S. Krol |
Title Awaited |
M.S. Shekhani |
Using
Sugars in Drug Discovery |
E. Carrier |
Artificial
Hematopoietic Stem Cell Niche Sustains Growth and Differentiation
of Human ES-Dervied Early Hematopoietic Pregenitors |
Y. Kitade |
Synthesis
of 2', 5' -Oligoadenylates Having Aromatic Groups and
their Biological Activities |
S. Dastmalchi |
Prediction
of Structural Features of Integral Membrane Proteins |
I.A. Bashir |
The
use of gum arabic fraction for treatment of chronic renal
failure patients |
A. Khalid |
From
Molecular Recognition to Drug Design:Applications of Experimental
and Theoretical Enzyme Inhibition Studies |
K. Fox |
Towards the Targeted Modulation of Gene Expression by
Modified Triplex-Forming Oligonucleotides |
K. Suzuki |
Protein
C Inhibitor Regulates Breast Cancer Cell Growth, Metastasis
and Angiogenesis |
F. Vallette |
Apoptosis
as a Target for Peptide and Protein Therapies |
A. Al-aboudi |
Cholinesterases
Inhibitory Activity of Testosterone and Some of its Metabolites |
M.A. Eldaway |
Design Studies of Drugs for the Management of Certain
Parasitic and Hepatic Viral Infections |
C.W. Huck |
Title Awaited |
B. Coulombe |
Inhibitors of Multisubunit RNA Polymerases as Tools to
Study Transcriptional Mechanisms in Prokaryotes and Eukaryotes |
A.H. Al-Marzouqi |
Effect
of Preparation Method on Physicochemical Properties of
Antifungal Drug-Cyclodextrin Complexes - Comparison between
Supercritical Carbon Dioxide and Conventional Methods |
C. Berthelette |
Case
Study of DP Receptor Antagonists: From HTS to Synthesis
and Selection of Pre-Clinical Candidate Compounds |
J. Bandow |
Identification
and Characterization of Novel Antibiotic Targets |
C.-H. Lai |
The
Asian Gynecologic Oncology Group and Clinical Trial Center
of Chang Gung Memorial Hospital |
H. Gardsvoll |
Mapping
Structural and Functional Epitopes for Ligand and Monoclonal
Antibody Binding on the Receptor for Urokinase-Type Plasminogen
Activator: Identification of Potential Target Sites for
Antagonist-Based Cancer Therapy |
V. Gault |
GIP-Based Therapeutics for Diabetes and Obesity |
A. Kamel |
The
Role of Aldehyde Oxidase in the Metabolism of the Antipsychotic
Drug Geodon |
H. Hassan |
Regioselective
Synthesis of Symmetric Pyridine-Spaced Sulfated Glucuronic
Acid and Study of Their Antiproliferative Activity |
A. Martinez |
From
Rational Drug Design To Disease Modifying Drugs For Alzheimer´s
Disease |
J. Chin-Dusting |
The
Heterogeneity of High Density Lipoproteins: Implications
for Therapeutic Development. |
C.-H. Chen |
New
Drug Development following Characterization of a Novel
Atherogenic Lipoprotein |
C. Szabo |
Development
of Gaseotransmitters (Nitric Oxide, Carbon Monoxide, Hydrogen
Sulfide) as Pharmaceutical Agents: Past Challenges, Future
Opportunities |
K. Ogata |
Regulatory
Mechanism of Assembly of Transcription Factors on DNA |
G. Kleymann |
Discovery
of New Drugs and Innovative Therapeutic Principles for
Superior Treatment of Herpes Disease |
P. Yu |
Vascular
Surface Semicarbazide-Sensitive Amine Oxidase (SSAO/VAP-1)
as a Novel Target for Treatment of Chronic Vascular Disorders
Associated with Protein Misfolding and Inflammation |
R. Alany |
Corneal
Delivery and Stability of Connexin 43 Antisense Oligonucleotides |
S. Al-Assaf |
Controlling
the Physicochemical Properties of Polysaccharides and
Proteins |
J. Blanchfield |
The
Development of Polymer Based Synthetic Vaccines |
J. Du Plessis |
Transdermal Delivery of Arginine Vasopressin with Pheroid™
Technology |
R. Falconer |
Selective
Delivery of Anti-Tumour Agents via Matrix Metalloproteinase
(MMP)-Cleavable Peptides |
M. Foldvari |
Prospects
for Non-Invasive Delivery of Proteins and Nucleic Acids
Across the Skin |
S. Celikoglu |
A
New Paradigm for Cancer Chemotherapy: Intratumoral Drug
Delivery |
M. Kuzuya |
A
Novel Drug Engineering by Plasma Technique |
R. Pasqualini/W. Arap |
Ligand-Directed
Therapy and Molecular Imaging based on In Vivo Phage Display
Technology |
K. Pankiewicz |
NAD-based
Anticancer Therapeutics |
M.A. Abdullah |
Cell
Engineering and Molecular Pharming for Biopharmaceuticals |
M. Walter |
High
Throughput X-ray Crystallography: Feeding the Drug Discovery
Pipeline |
Z. Witczak |
Thio-sugars
as Emerging Targets for Carbohydrate Therapeutics Discovery |
T. Al Tel |
Diversity-Oriented
Synthesis: Enantioselective Synthesis of a Pool of Small
Molecules as Drug Candidates |
A. Peracchi |
How (and why) to revive a dead enzyme: the power of
chemical rescue |
N. Zgheib |
The
Effect of Liver Disease on Cytochrome P450 Mediated Metabolism |
V. Brabec |
Platinum
Coordination Complexes. from DNA Interactions to New Anti-Tumor
Drug Design |
I. Gockel |
Novel
Therapeutic Targets in Esophageal Cancer: Impact of Coexpression
of Receptor-Tyrosine-Kinases (RTK) and Chemokine Receptor
CXCR4 |
R. Kiss |
The
Sodium Pump and Its Alpha1 and Alpha3 Subunits as Novel
Targets to Combat Apoptosis- and/or Multidrug-Resistant
Proliferating and Migrating Cancer Cells |
V. Djonov |
Title Awaited |
A. Pertis |
Non-Natural Nucleotide Analogs as Probes of DNA Polymerase
Activity |
A. Ali |
Discovery
of Novel, Selective Glucocorticoid Receptor Modulators |
R. Assaly |
Plasma
Expansion by Polyethylene Glycol Modified Albumin (PEG-Alb) |
L. Chugh |
Dengue
Virus Viremia: Role of NS1 Protein of Virus / Cytotoxic
Factor Produced by T-Cells |
J. De Sanctis |
New
Glutarimide Alkaloids as Potent Anti-Inflammatory Drugs |
C.D. Ribas |
Relevant Effects of Omalizumab, an Anti-Ige Drug, In Asthma
and other Diseases |
P. Sayeski |
Jak2 and Reactive Oxygen Species: A Complex Relationship |
G. Leclercq |
Implication
of Estrogen Receptor α
in Breast Cancer Development - A New Concept for the Development
of Drugs Aimed to Antagonize its Action |
C.-T. Lin |
Peptide-Targeted
Chemotherapy against Nasopharyngeal Carcinoma |
S. Linder |
A
Biomarker Concept for Anticancer Drug Development |
N. Eikje |
Identification
and Characterization of Skin Biomolecules for Drug Targeting
by Vibrational Spectroscopy |
Y.-C. Kuo |
The
Immunomodulatory Activities of (S)-Armepavine on Autoimmune
Diseases In vivo and In vitro |
W. Chegwidden |
The
Carbonic Anhydrases: Potential Therapeutic Targets in
Renal Carcinoma |
G.B. Fields |
Mechanism
and Inhibition of Collagenolytic Matrix Metalloproteinases |
S. Qureshi |
Improved In vitro Model to Assess Drugs Release
Characteristics of Products for their Absorption from
Human Gastrointestinal Tract |
B. Imbimbo |
The
Therapeutic Potential of γ
-Secretase Modulators in Treating Alzheimer’s disease |
M. Botta |
The
Fight against AIDS: New Avenues for Inhibiting RT, an
Old Target |
T. Prisinzano |
Discovery
of mu Opioids with altered Receptor Regulation |
N. Zawia |
A
Novel class of Mechanism-based Drugs for the Treatment
of Alzheimer’s Disease |
U. Holzgrabe |
Piggy
Back Approach: Bisaphthalimides As Muscarinic Agnoists,
Cancerostatics, And Antiinfectives |
R. James |
Developing
Novel Antimicrobial Peptides Active Against Gram-Positive
Pathogens |
L. Polonelli |
Engineered
Antibody Cdrs As Novel Antimicrobial, Antiviral And Antitumor
Drugs |
C. Salmi |
Squalamine,
A New Antibiotic Extracted From Marine Environment: How
about Its Mechanism Of Action With Respect to Gram-Negative
Bacteria? |
M. Alam |
High
Throughput Compound Library Screening for Potential Antiviral
Drugs for Dengue Virus |
K.-I. Sato |
Focused
Proteomics on Membrane Microdomain-associated Signal Transduction
in Fertilized Amphibian Eggs and Human Bladder Carcinoma
Cells |
P. Aljama |
Optimizing
the Use of Erythropoiesis Agents (ESA) in Renal Anemia |
A. Pini |
Identification,
Optimization and In vivo Activity of a Branched
Antimicrobial Peptide Selective For Gram-Negative Bacteria |
H.-M. Chen |
Structure
of a Novel Anticancer Peptide CB1a, Based on the N-terminal
Peptide Sequence of Cecropin B |
L.-K. Chau |
Rapid
and Label-Free Bio-Detection Based on Localized Plasmon
Resonance |
D. Steinbach |
Which
ABC-transporters should we target in Leukemia? |
E. Terpos |
Proteasome
Inhibition Therapies and Bone Metabolism in Multiple Myeloma |
M. Turkay |
Identification
of Drug Candidates for Prostate Cancer Using Computational
and Experimental Methods |
S. Shigeta |
Anti-RNA
Virus Activity of Polyoxometalates |
D. Buchi |
Immune
System Modulation with a Homeopathic Medication. |
W. Childers |
Serotonergic
Drug Design - Finding Diamonds in the Rough |
Y. Collette |
HIV-1
nef-SH3 Targeting as a Proof of Concept for the Development
of Anti-Viral Protein-Protein Interaction Inhibitors |
E. Elzein |
Discovery
of CVT-6883: A Novel A2B Adenosine Receptor Antagonist
as a Clinical Candidate for the Treatment of Asthma |
A. Grobler |
Pheroid
TM Technology: A Novel Drug Delivery System with Broad
Application |
B.Noszal |
Molecular
Mechanism of Morphine-6-Glucuronidate Brain Penetration |
J.O.V. Planells |
Transcorneal Permeation of Nsaids Drug Delivery in a Corneal
Device |
S.E. Mansour |
Synthesis
and Antimicrobial Activity of some Novel Oxadiazole Derivatives |
A. Damas |
TTR
Amyloidosis: from the Molecular Mechanism to Therapy |
K. Filipiak |
How
can we Prevent Diabetes in Pharmacological way ? |
H. Kang |
Peroxisome
Proliferator-Activated Receptor Delta Selective Agonists
as Potent Anti-Atherogenic Agents In vivo |
J. Zablocki |
Novel
Aldehyde Dehydrogenase-2 Inhibitors as a Potential Treatment
of Alcohol Addiction |
C. Assaf |
Emerging
Drugs in Cutaneous Lymphomas |
S. Kumar |
Can
the Acute Toxicity of Antidepressants be Predicted Using
the Protozoan Tetrahymena pyriformis? |
D. Dizon |
From
Bench to Bedside: The clinical development of pertuzumab
in women's cancers |
M. Gyongyossy-Issa |
A
synthetic platelet as application of a targeted controlled-rate
drug delivery vehicle |
H.-G. Ljunggren |
Prospects
for the Use of NK-Cells in Immunotherapy Against Human
Cancer |
G.-J. Wang |
Endotoxin-Stimulated
Responses and Therapeutic Herbal Medicines Development
by a Systems Biology Approach |
M.J. Drysdale |
Structure
Based Discovery of Hsp90 Inhibitors for the Treatment
of Cancer |
B. Ahmed |
Antihypertensive, Cardiovascular and β-Blocking
Adrenergic Activity of Aryloxypropanolamines |
A. El-Dahshan |
An
Efficient Solid Phase Synthesis Concept for the Preparation
of various Novel Biologically Active Peptide Mimetics |
E. Goldsmith |
Unique
Autoinhibitory Dimers in the MAP2K MEK6, and MAP4K OSR1 |
R. Scott |
Title awaited |
M. Shamssain |
Novel
Strategies for the Treatment of Asthma and COPD - Future
Challenges of Drug Therapy |
H.H.A.-M. Hassan |
Regioselective
Synthesis of Symmetric Pyridine-Spaced Sulfated Glucuronic
Acid and Study of their Antiproliferative Activity |
R. Howes |
Development of Inhibitors of Hsp90 for Cancer Therapy:
The Screening Story |
Name of Presenter |
Title |
E. Afrasiabi |
Anticancerous
Properties of Phorbol 12-Myristate 13-Acetate (PMA) in
Human Thyroid Cancer Cells |
Z. Zaheer |
Stability
indicating HPTLC Determination of-Carvedilol in Pharmaceutical
Dosage Form |
P. Alexandrino Fernandes |
Computational
Mapping of Druggable Sites in Proteins |
M. Abdouss |
Uniformly
Sized, Molecularly Imprinted Polymers for Enantioselectivity
of Pseudoephedrine by Precipitation Polymerization |
P. Andrade |
HPLC-DAD-MS/MS-ESI
Screening of Phenolics with Potential Bioactivity in Pieris
Brassicae L. Reared on Brassica Rapa Var Rapa L. |
M. Alam |
High
Throughput Compound Library Screening and Herbal Supplements
to Mitigate Dengue Fever |
N.A. Atatreh |
Inhibition
of Src for Potential Use in Cancer Chemotherapy |
A.M. Aubertin |
Anti-HIV
Prodrugs Conjugating a Reverse Transcriptase Inhibitor
with Integrase Inhibitors by a Spontaneously Cleavable
Linker: Synthesis and Evaluation of Antiviral Activity |
M. Beiner |
Nanoconfinement:
A strategy to manipulate the crystallization behavior
of drugs |
N. Belacel |
Intelligent
Decision Support System-Based Biomarker Discovery |
K. Orrling |
Investigation
of the P1’ Substituent - Synthesis and Evaluation
of Inhibitors of Malarial Aspartic Proteases. |
L. Navidpour |
Synthesis
and Anti-helicobacter Pylori Activity of (Z)-2-(nitroimidazolylmeth-
ylene)-2(3H)-Benzofuranone Derivatives |
M. Asahi |
Discovery
of a Drug that Blocks the Trojan Horse-like Strategy Used
by Pathogenic Helicobacter pylori and its Associated Bacteriophage |
Y.-an Bi |
Use
of the Cryopreserved Human Hepatocyte Sandwich-Culture
Model to Measure Hepatic Metabolism and Biliary Efflux |
D. Bikiaris |
Improvement
of Fluvastatin Controlled Release Through the Use of New
Biocompatible Aliphatic Polyesters |
L. Krivankova |
Elimination
of Matrix Effects in Analyses of Trace Metabolites in
Body Fluids by Capillary Electrophoresis |
G. Horvath |
Synthesis,
Characterization, and Biomedical Evaluation of a Novel
Water-Soluble Platinum-Based Anticancer Drug |
N. Bovin |
New
Paradigm in Anti-Viral Therapy |
J. Breytenbach |
1.
Cytarabine Prodrugs for Transdermal Delivery 2.
Novel Prodrugs of Lamivudine and Zidovudine for Transdermal
Delivery in the Treatment of HIV/AIDS |
F. Burczynski |
Hepatoprotective
Effect of Diltiazem and Silymarin. |
F. Carrier |
Molecular
Understanding of Histone Deacetylase Inhibitors (HDACIs)
Efficiency in Cancer Cells. |
L. Chalissery |
An
Effective Purification Method for Cucurbit [N]Uril; A
Molecular Host and Drug Delivery Vehicle |
M. Furch |
Allosteric
Inhibitors of Myosin Function |
J. Du Plessis |
Transdermal
Delivery of Arginine Vasopressin with Pheroid™ Technology |
A. Chimirri |
Combined
Ligand-Based and Target-Based Approach to Design NR2B/NMDA
Receptor Antagonists |
J. Chin |
A
Semi-Total Synthesis of Guggulsterones, Natural Hypolipidemic
Drugs, from Various Steroids |
C. Soria |
A
Novel Strategy of Anti Cancer Therapy: Targeting Specifically
the Gtpase Rhoa and Development of a New Strategy for
Sirna Therapy: In Vitro and In Vivo Assays |
S. Christensen |
Peptide
Inhibitors of DNA Replication in Staphylococcus Aureus |
S. Achour |
Kinetic
study on the Decomposition of 2-Chloroethylnitrososulfamides
(CENS) in Organic Media |
E. Valeur |
Dual
Fragment Microarrays : Towards a New Perspective for Drug
Discovery |
M. Correia-da-Silva |
Anticoagulant
Actions of Structure-Diverse Sulfated Phenols |
R. Dghaim |
Palladium
Catalyzed Multicomponent Reactions: A Facile One-Pot Coupling
Approach to α-Amino
Acid and Peptide Derivatives |
H. Doi |
Pd(0)-Mediated
Rapid C-Methylations for the Synthesis of 11C-Incorporated
PET Tracerrs |
G. Duburs |
Peptide-Like
and Lipid-Type Compounds on the Basis of Unsaturated Cyclic
Amino Acids-Carbonyldihydropyridines |
H. Durchschlag |
Modeling
of Individual Water Molecules Preferentially Bound to
Proteins |
D. Egan |
Apoptotic
Cell Death and Cell Cycle Events Mediate the Action of
6-Hydroxycoumarin-3-Carboxylatosilver in Human Malignant
Hepatic Cells |
B. Flynn |
Discovery
of BNC105P, A Clinical Candidate for the Treatment of
Cancer: A Case Study in the Application of the Diversity-Oriented
Synthesis Technology, MultiCore® |
E. Fagadar-Cosma |
New
Asymmetric meso-Tetraphenylporphyrins Peripherally Diverse
Substituted with Pyridyl or Dimethoxy Groups as Promising
Photosensitizers in Photodynamic Therapy |
A. Siriviat |
Electric
Field Drive Transdermal Drug Delivery of Salicylic Acid
-Loaded Polyacrylamide Hydrogels |
I.M. Fenyo |
Retinoids
Induce Apoe Gene Upregulation in Macrophages |
P. Kothary |
Greater
Inhibition of Connective Tissue Growth Factor Synthesis
By a MAP Kinase Inhibitor Compared to Amino Guanidine
in Cultured Human Retinal Pigment Epithelial Cells |
S. Gobec |
New
Inhibitors of D-Alanine:D-Alanine Ligase (Ddlb) Discovered
By Structure-Based Virtual Screening of the NCI Diversity
Set |
K. Goracinova |
Efficacy
of Microparticulated Bds Dosage Forms in the Treatment
of Experimentally Induced Colitis in Rats |
T. Kowalska |
On
the In Vitro Oscillatory Chiral Inversion of
Selected L-Amino Acids and its Implications. |
K. Shayesteh |
Powder
Mixing and Influence of Solvent on Mixture Quality in
the Production of Amlodipin Tablet |
H.R. Ha |
Chemical
Structure-Aqueous Solubility Relationship of Amiodarone |
G. Hadzic |
Dynasore is not Dynamin Inhibitor |
V. Khavinson |
Peptide
Regulation of the Functional Activity of the Retina |
E.W. Hansen |
A
Novel Human-Cell Based Pyrogen Test |
R. Akkina |
A
New Humanized Mouse Model for Testing HIV/AIDS Therapies
and Microbicides |
M.Y. Yoon |
Overexpression
of Tubulin and its Inhibitor Screening for Microtubule
Formation in Phytophthora Capsici |
M. Hassan |
Antineoplastic
Effects of α-Terpineol,
Linalyl Acetate and dl-Camphor, Components of Lebanese
Sage Essential Oil |
R. Ward |
Correlation
of Activity and Sequence Similarity in Kinase Targets |
S. Hassan |
Antineoplastic
Effects of α-Terpineol,
Linalyl Acetate and Dl-Camphor, Components of Lebanese
Sage Essential Oil |
K. Musilek |
Acetylcholinesterase
Reactivator – Oxime HI-6 – Antidote Against
Nerve Agents |
H. Hibasami |
Blazein
(A New Steroid) Isolated from Mushroom (Agaricus blazei
Murill) Induce Apoptosis in Human Lung Cancer LU99 and
Stomach Cancer KATO III Cells |
T. Bruckdorfer |
PEGylation
– A Key Technology to improve Solubility and Pharmacokinetic
of Peptides, Proteins and other Biopharmaceuticals for
Superior Drug Delivery |
M. Steiert |
Nanoparticle-Based
Delivery of Aminoglycoside Antibiotics |
S. Imreh |
A
Microcell Hybrid Based "Elimination Test" in
Anticancer Drug Design |
D. Janezic |
Protein-Protein
Binding Sites Prediction |
G.A. Spyroulias |
Novel
Insights into Angiotensin-Converting Enzyme Domain Selectivity
& Structure-Based Drug Design |
K. Al-Kuraya |
Ubiquitin-Ligase SKP2 Pathway is an Attractive Target
for Colorectal Cancer Therapy |
A. Helgee |
A
Method for Automated Molecular Optimization by Inverse
QSAR Applied to Ames Mutagenicity Data |
R. Kamel |
Polymeric
Matrix System for Transdermal Delivery of Tramadol Hydrochloride |
S. Kanan |
Detection
and Identification of Banned Chemicals in Dietary Food
Supplements |
E. Karavas |
Hydrogen
Bonding Interactions as a New Sustain Release Mechanism |
J. Kasparkova |
Unique
Properties of DNA Interstrand Cross-Links of Antitumor
Oxaliplatin |
J. Kelly |
Can
the Acute Toxicity of Antidepressants be Predicted Using
the Protozoan Tetrahymena pyriformis? |
A. Sirivat |
Controlled
Release of Sulfosalicylic Acid from Polypyrrole/Poly(acrylic
acid) Hydrogel by Electrical Stimulation |
J. Garmendia |
β2
Adrenoreceptor Polymorphism in Asthmatic Population in
Venezuelan |
A. Khvat |
Rational
for Focused DiversityTM Approach to Discovery of Signaling
and Developmental Pathway Inhibitors. A Case Study for
PI3K and Hh Modulators |
L. Carlsson |
Local
Interpretation of Machine-Learning Models using Attribute
Gradients, Applied to Ames Mutagenicity Data |
P. Ohrngren |
Evaluation
of Various P1’ Substituents in Tertiary Alcohol
Containing and Elongated HIV-1 Protease Inhibitors |
O. Lagerlund |
α-Arylation
of a Protected Glycine in Water: 3-Phenylglycine Derivatives
as Inhibitors of the Tuberculosis Enzyme, Glutamine Synthetase |
L. Kock |
Aspirin:
The Anti-Inflammatory Antifungal |
A. Vakili |
Effect
of central blockage of gap junction by Carbenoxolone on
ischemic damage in transient model of focal cerebral ischemia |
S. Komba |
General
Strategy for Synthesis of Oligosaccharide Combinatorial
Library to Develop for Oligosaccharide Array |
H. Fessi |
Preparation
and Characterization of Radioactive Dirhenium Decacarbonyl-Loaded
PLLA Nanoparticles for Radionuclide Intra-Tumoral Therapy |
E. Valeur |
Towards
Potent Inhibitors of the Mdm2-P53 Protein-Protein Interaction |
J.S. Kovach |
A
New Inhibitor of Serine-Threonine Protein Phosphatase,
PP2A, Suppresses
Growth and Induces Differentiation of Medulloblastoma
Cells |
M. Asahi |
Therapy
against Microbial-Encoded ITAM-Like Motifs May Treat and/or
Prevent a Number of Serious Infections Caused by Microbial
Pathogens |
M. Kukhanova |
Design
of Depot Forms of Anti-Hiv Agents Based on Nucleoside
-Phosphonate Derivatives |
G. Kulcsar |
Preclinical
Experiments on Culevit Infusion Developed on the Basis
of a Passive Antitumor Defence System and Investigation
of Mechanism |
K.L. Lou |
Improvement
of Drug Virtual Screen By GA/GP: Docking Studies on Tubulin
Inhibitors as Anticancer Agents |
B. Lammek |
Influence of Bulky 3, 3- Diphenylalanine Enantiomers
Replacing Position 2 of Arginine Vasopressin and its Analogues
on their Pharmacological Properties |
E. El-Bastawiss |
Molecular
Docking and Analysis of Certain Potent Anti-angiogenic
Vascular Endothelial Growth Factor Receptor-2 (VEGFR2)
Inhibitors |
F. Lefranc |
Narciclasine
Displays Potent and Selective Anti-Tumor Effects by Impairing
Cancer Cell Migration Through a Phosphocofilin-Mediated
Increase of Actin Stress Fibers |
W. Liebenberg |
An
In vitro Evaluation of the Efficacy of Anti-Malaria Drugs
by Pheroid™ Technology |
J.C. Lin |
Inhibitory Effects of Some Derivatives of Glycyrrhizic
Acid against Epstein-Barr Virus Infection: Structure-Activity
Relationships |
M. Lise |
Effect
of Moist Heat Sterilisation on Pyrogenicity of Whole Bacteria
and Cell Wall Components from Staphylococcus aureus |
Z. Zidek |
Novel
Group of Biological Response Modifiers: Inhibitors of
Endoplasmic Ca2+-ATPase |
A.A. Taherian |
Comparison
the effects of aqueous extract of Glycyrrhiza Glabra,
Dexamethasone and stress on acute and chronic pains in
mice |
M. Degani |
Synthesis
and Biological Evaluation of Novel Antifolates Towards
Filariasis |
Y. Zhao |
Cucurbit[N]
Uril for Drug Delivery |
A. Maghazachi |
The
Copolymer-1 Glatiramer Acetate (Copaxone) Inhibits Natural
Killer (NK) Cells Lysis of Tumor Cells but Enhances Their
Cytolysis of Syngeneic or Allogeneic Immature and Mature
Monocyte-Derived Dendritic Cells |
R. Müller |
Action of Disorazol A in Combination with Other Tubulin-active
Compounds |
N. Belacel |
Theoretical
Analysis of Metabolic Pathways in Cancer Development -
The Effect of Zn2+ Concentration Changes on
Prostate Cell Metabolism - Authored by Miroslova Cuperlovic-Culf
and Nabil Belacel |
B. Zhang |
In
Silico Protein-Protein Interaction Peptide Inhibitors
Design for Cyclin-Dependent Kinase5 (CDKs) |
M.C.Manca de Nadra |
Viability
Modification of Listeria Monocytogenes by the Effect of
Phenolic Compounds Combination |
J. Bappu |
A
Novel Therapeutic Use of Fibrin Sealant to Promote Saphenous
Graft Wound Healing in Patients Undergoing Cardiac Surgery:
A Randomised Study |
A. Khalid |
Searching
for New Cholinesterases Inhibiting Drug Candidates from
Natural Sources |
A. Yarat |
Investigation
of the Effect of Silymarin on the Liver in Experimental
Sepsis |
E. Mohamed |
Probing
the HIV Reverse-Transcriptase Enzyme: Synthesis and Biological
Evaluation of Novel Bifunctional NRTI/NNRTI HIV-1 Reverse-Transcriptase
Inhibitors |
A. S. Yang |
Molecular Modeling of Protein-Substrate Interactions
in Factor-Xa with High-Throughput Substrate Phage-Display
Data |
M. Muñoz |
Neurokinin
1 Receptor Antagonist Aprepitant as an Antitumor Drug |
P. Muretto |
Endogastric
Capsule for E-Cadherin Gene (CDH1) Promoter Hypermethylation
Assessment in DNA from Gastric Juice of Patients with
Gastric Cancer |
A. A. Vafaei |
Effect
of hydro-alcoholic extract of Valeriana Officinalis on
Anxiety related behavior in mice: An interaction with
Serotonergic and Noradrenergic systems |
S. Shen |
Preparation
and Characterization of (3-aminopropyl)triethoxysilane-Modified
Silica Nanoparticles for Protein Delivery |
N. Nifantiev |
Phenolic
Compounds From Siberian Conifer Trees – Multi-Purpose
Drug Substances and Functionalized Scaffolds for Nces
Design |
M. Noguchi |
Combination
Therapy of Personalized Peptide Vaccination and Low-Dose
Estramustine Phosphate for Metastatic Hormone Refractory
Prostate Cancer Patients |
A. Rashidy-Pour |
Post-training
administration of corticosterone enhances consolidation
of contextual fear memory and hippocampal long-term potentiation
in rats |
I. Tvaroska |
Design
and Synthesis of Transition State Inhibitors for Glycosyltransferases |
D. Tweedie |
Orally
Active TNF-Alpha Synthesis Inhibitors: A Role in the Treatment
of Neurodegeneration? |
R. Ondarza |
Novel
Anti-Parasitic Targets from Human Pathogenic Amoebas:
Entamoeba histolytica, Acanthamoeba Polyphaga and Naegleria
fowleri |
S. Oniga |
Synthesis
of Some New Hydrazino-Thiazolic Compounds |
M.d. Palage |
Synthesis
and Physicochemical Characterization of Some Thiazolium
2-Aryl Ammonium Quaternary Salts |
E. Topic |
Pharmacogenetic
Approaches in Psychiatric Patients |
M. K. Park |
An
Anticancer Peptide Histonine Derived from Histonine H2A
and its Mechanism of Action |
S. H. Park |
The
Absorption, Distribution, Excretion and Pharmacokinetics
of Carbon-14 Labeled Pyronaridine Tetraphosphate in Sprague-Dawley
Rats |
B. Tiperciuc |
The
Effect of Some New Synthesis Flavonoids on Inflammation-Induced
Oxidative Stress |
J. Hirsch |
Nanoparticle-Based
Delivery of Aminoglycoside Antibiotics |
A. Parvu |
The
Effect OF Some New Chromanon-1,3,4-Oxadiazolines on Inflammation-Induced
Nitric Oxide Synthesis |
D. Patinkin |
The
Effect of Pegylated Antisense Acetylcholinesterase on
Hematopoiesis |
J.U. Peters |
NK1
/ NK3 Dual Antagonists: Finding a Lead for a Schizophrenia
Drug Discovery Programme |
M. Pinto |
Prenylation
on Xanthonic and Flavonic Scaffolds: A Key Approach for
Antitumor Activity |
A. Poot |
Design
and Synthesis of Isozyme Selective Protein Kinase C Inhibitors |
M. Rosso |
Neurokinin
1 Receptor Antagonist Aprepitant as an Antitumor Drug |
T. Kowalska |
On
the in Vitro Oscillatory Chiral Inversion of Profen Drugs
and Its Implications |
Y. Takizawa |
Biochemical
Analysis of Two Isoforms of the Human Rad51 Protein |
M. Timm |
Cryopreservation
of Differentiated HL-60 Cells – Development of a
Novel in vitro Pyrogen Testing Kit |
S. Sharma |
Synthesis,
Biodistribution and Pharmacological Studies of Iozapine:
A Potential Ligand for Brain Imaging |
E.J. Sheridan |
Boronated Peptides for Boron Neutron Capture Therapy |
M.E. Sousa |
Antiproliferative
Effects and Enhancement of the Growth Inhibitory Action
of 4-Hydroxytamoxifen in Estrogen Receptor Positive (ER+)
Breast Cancer Cell Line Induced By Prenylated Xanthones |
G.A. Spyroulias |
A
Residue Specific Sight of Anthrax Lethal Factor –
Mkks Interaction and Selectivity Towards Structure-Driven
Drug Design |
V. Khavinson |
Molecular and Genetic Mechanisms of Effect of Peptide
Geroprotector Pharmaceuticals |
J.-L. Peglion |
Benzocycloalkane Derivatives as Potent Serotonin Reuptake
Inhibitors |
A.F. Faruqi |
The Synthetic Growth Surface Topography of Ultra-Web™
Enhances Hepatocyte Culture Performance Compared to Biological
Coatings |
C. Fernandez |
Synergistic
Application of NMR, MS and X-Ray for Fragment-Based Screening:
A Critical Assessment |
A. Kamel |
High
Throughput Sample Analysis for Identification and Quantitative
Assessment of Library Screening Using Ultra Performance
Liquid Chromatography/Ultra Violet/ Evaporative Light
Scattering Detection Coupled to Time of Flight Mass Spectrometry
(UPLC/UV/ELSD/TOFMS) |
C. Prakash |
Use
of the Cryopreserved Human Hepatocyte Sandwich-Culture
Model to Measure Hepatic Metabolism and Biliary Efflux |
A. Nicolin |
Increase BCl2 Expression by ssRNA Complementary
to the ARE Motif |
E. Sletten |
Cytotoxic Trans- platinum Iminoether Complexes form
Adducts only with Single-Stranded Oligodeoxynucleotides. |